平安! 发表于 2011-11-9 19:57
6 b# }8 y5 N+ F+ } G) F& H$ ]Pazopanib (100 mg/kg/day free base equivalent)
: g* i: x" H; T _9 U 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。$ j# U2 U" ]- @$ N2 C
搜索了一下,原料一大堆。
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" C- X, C8 }4 Z; }$ c/ j' s! V f对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。8 s( V$ F n% ~: E1 K+ t4 A0 l* n
% o. a% C6 g7 i- l- h--------------------- DOSAGE AND ADMINISTRATION ----------------
# o: W. t9 {* n# v* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
* _( A: ?: k0 l5 q6 f# G* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
( M6 U1 u) v" E% J, A---------------------DOSAGE FORMS AND STRENGTHS --------------5 j6 w C# ^' p
200 mg tablets. (3)
* l* ^+ \* T3 [3 m-------------------------------CONTRAINDICATIONS------------------------ |