平安! 发表于 2011-11-9 19:57 9 Y, l \5 Y5 i, N8 ] ~4 }; i4 U
Pazopanib (100 mg/kg/day free base equivalent) , N/ y4 ?/ B8 _1 u
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
* a8 I) B C% R' g搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。3 W7 k& |% Y' ^# s3 I1 e/ l
$ h7 y9 I {. `- Y2 B9 G以下是正版说明书的推荐用量。; g8 d+ [6 b+ T( Q4 M- c
+ d5 {, U# a/ f3 ~6 H--------------------- DOSAGE AND ADMINISTRATION ----------------5 b0 p, n# Y, W' C3 q
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
9 u, H! U; O, p$ F* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
8 p- G+ j( d3 Y4 [9 p---------------------DOSAGE FORMS AND STRENGTHS --------------
8 X6 N7 Y7 W1 ~$ V200 mg tablets. (3) 4 x; R' S2 ~9 T- o
-------------------------------CONTRAINDICATIONS------------------------ |