平安! 发表于 2011-11-9 19:57 8 }6 V7 P% {+ ~7 A7 M1 I
Pazopanib (100 mg/kg/day free base equivalent)
, e" J7 H' k# Y, I3 U4 P& ^! x 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
/ G$ q4 y! i8 c Z0 [# ^* m搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。, }5 P3 j5 N5 d: }8 d+ d
~3 |' y. ~4 w( N3 H# Q, s' l以下是正版说明书的推荐用量。
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s& i- z* J# B--------------------- DOSAGE AND ADMINISTRATION ----------------
5 w5 Z" G0 b; n5 ^9 I8 t6 t) C* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
& P6 t5 h* A* e1 n, n% f6 f% x* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
7 p4 N4 h, ?7 X% h+ H* J1 N---------------------DOSAGE FORMS AND STRENGTHS --------------7 X/ P/ i- m3 y+ h3 G: q
200 mg tablets. (3)
% _1 O$ R# v5 o# l0 I. E-------------------------------CONTRAINDICATIONS------------------------ |