平安! 发表于 2011-11-9 19:57
( w) q, u+ \* M* T3 L: lPazopanib (100 mg/kg/day free base equivalent)
! S. B4 O, q- j4 h6 A 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
- X" b6 k$ i K搜索了一下,原料一大堆。& R0 |0 S0 u; A3 N+ z9 G
2 R" [0 q" }) U* m% Q对不起!100mg/kg是用于移植瘤的,我弄错了。
$ z [3 a' a/ d9 K7 h' n4 ^; [/ {0 C8 e) |3 k/ p- w
以下是正版说明书的推荐用量。0 {0 O0 F- D8 O: J# Z
" t" H3 k$ D e9 M. _8 N--------------------- DOSAGE AND ADMINISTRATION ----------------/ E! }9 c# F8 e9 P) `* D1 _
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
' N" O- e# j' \0 K0 J, i) C7 L* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
9 L L4 O, ]" F# R( s---------------------DOSAGE FORMS AND STRENGTHS --------------- I0 ^( P! q2 D
200 mg tablets. (3) 9 P+ p! \/ a. N+ M1 {; X4 a( a9 G
-------------------------------CONTRAINDICATIONS------------------------ |